4-Tert-butylbenzene-1,2-diamine → HCID 178440695, compound

HRID 1424169Notes

Reaction equation

HRID 1424169 reaction equation
C(OC([N:8]1[C@@H:14]([C:15](O)=O)[CH2:13][CH2:12][CH2:11][O:10]C1(C)C)=O)(C)(C)C.[C:20]([C:24]1[CH:29]=[CH:28][C:27]([NH2:30])=[C:26]([NH2:31])[CH:25]=1)([CH3:23])([CH3:22])[CH3:21]>>[NH2:8][C@@H:14]([C:15]1[NH:30][C:27]2[CH:28]=[CH:29][C:24]([C:20]([CH3:23])([CH3:21])[CH3:22])=[CH:25][C:26]=2[N:31]=1)[CH2:13][CH2:12][CH2:11][OH:10]

Participants

3

Reactant 2

HCID 4327084-Tert-butylbenzene-1,2-diamineHCID 86699071HCID 86699071, compound

Product 1

HCID 178440695HCID 178440695, compound

Procedure

The title compound was prepared according to Method 4 using (4R)-3-(tert-butoxycarbonyl)-2,2-dimethyl-1,3-oxazepane-4-carboxylic acid (Preparation 48) and 4-tert-butyl-1,2-diaminobenzene.

Sources & evidence

ORD record
ord-59512f1e96754338bd93ebccd56693fd
Source dataset
uspto-grants-2015_01
Patent number
US08927587B2

Reaction notes

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