(6-Methoxy-1-benzothiophen-2-yl)boronic acid → HCID 57936114, compound

HRID 1434969Notes

Reaction equation

HRID 1434969 reaction equation
[CH3:1][O:2][C:3]1[CH:4]=[CH:5][C:6]2[CH:10]=[C:9](B(O)O)[S:8][C:7]=2[CH:14]=1.Cl[C:16]1[CH:21]=[CH:20][N:19]=[C:18]([NH:22][CH:23]2[CH2:28][C:27]([CH3:30])([CH3:29])[NH:26][C:25]([CH3:32])([CH3:31])[CH2:24]2)[N:17]=1>>[CH3:1][O:2][C:3]1[CH:4]=[CH:5][C:6]2[CH:10]=[C:9]([C:20]3[CH:21]=[CH:16][N:17]=[C:18]([NH:22][CH:23]4[CH2:28][C:27]([CH3:30])([CH3:29])[NH:26][C:25]([CH3:32])([CH3:31])[CH2:24]4)[N:19]=3)[S:8][C:7]=2[CH:14]=1

Participants

3

Reactant 2

HCID 10560276(6-Methoxy-1-benzothiophen-2-yl)boronic acidHCID 57936167(4-Chloro-pyrimidin-2-yl)(2,2,6,6-tetramethyl-piperidin-4-yl)-amine

Product 1

HCID 57936114HCID 57936114, compound

Procedure

The title compound was prepared analogous to Method C, starting 6-methoxy-benzo[b]thiophen-2-boronic acid and (4-Chloro-pyrimidin-2-yl)-(2,2,6,6-tetramethyl-piperidin-4-yl)-amine.

Sources & evidence

ORD record
ord-edced1b9056c4ccb906546d71c28cf33
Source dataset
uspto-grants-2009_11
Patent number
US07615562B2

Reaction notes

Loading…