4-Amino-2,2,6,6-tetramethylpiperidine → HCID 57936154, compound

HRID 1434974Notes

Reaction equation

HRID 1434974 reaction equation
[CH3:1][O:2][C:3]1[CH:4]=[CH:5][C:6]2[CH:10]=[C:9](B(O)O)[S:8][C:7]=2[CH:14]=1.Cl[C:16]1[N:21]=[C:20](Cl)[C:19]([CH3:23])=[CH:18][N:17]=1.[NH2:24][CH:25]1[CH2:30][C:29]([CH3:32])([CH3:31])[NH:28][C:27]([CH3:34])([CH3:33])[CH2:26]1>>[CH3:1][O:2][C:3]1[CH:4]=[CH:5][C:6]2[CH:10]=[C:9]([C:18]3[C:19]([CH3:23])=[CH:20][N:21]=[C:16]([NH:24][CH:25]4[CH2:26][C:27]([CH3:34])([CH3:33])[NH:28][C:29]([CH3:32])([CH3:31])[CH2:30]4)[N:17]=3)[S:8][C:7]=2[CH:14]=1

Participants

4

Reactant 3

HCID 375244-Amino-2,2,6,6-tetramethylpiperidineHCID 74508Pyrimidine, 2,4-dichloro-5-methyl-HCID 10560276(6-Methoxy-1-benzothiophen-2-yl)boronic acid

Product 1

HCID 57936154HCID 57936154, compound

Procedure

The title compound was prepared analogous to Method A, starting 6-methoxy-benzo[b]thiophene-2-boronic acid, 2,4-dichloro-5-methyl-pyrimidine and 4-amino-2,2,6,6-tetramethylpiperidine.

Sources & evidence

ORD record
ord-6aabb7abfcb64fa7b4c28ce28393746d
Source dataset
uspto-grants-2009_11
Patent number
US07615562B2

Reaction notes

Loading…