Potassium Carbonate → HCID 11661891, compound

Participants

Reaction Steps

Prepare using the method of Example 103 with palladium (II) acetate (0.002 g, 0.008 mmol), anhydrous acetonitrile (4 mL), triphenylphosphine (0.009 g, 0.034 mmol), distilled water (1 mL), 4-(methanesulfonyl)benzeneboronic acid (0.096 g, 0.45 mmol), 2-(4-bromophenyl)-4-{2-[(3S)-3-fluoropyrrolidin-1-yl]ethyl}-5-methyl-1,3-oxazole (See Example 104) (0.150 g, 0.42 mmol) and potassium carbonate (0.176 g, 1.27 mmol) to give the title compound as a cream coloured solid (0.133 g): MS (m/e): 429(M+1).

Provenance & Evidence