Potassium Carbonate → HCID 11676556, compound

Participants

Reaction Steps

Prepare using the method of Example 103 with palladium (II) acetate (0.003 g, 0.015 mmol), anhydrous acetonitrile (4 mL), triphenylphosphine (0.016 g, 0.059 mmol), distilled water (1 mL), 4-(methanesulfonyl)benzeneboronic acid (0.24 g, 1.11 mmol), 2-(4-bromophenyl)-4-{2-[(3S)-3-methoxypyrrolidin-1-yl]ethyl}-5-methyl-1,3-oxazole (See Example 117) (0.27 g, 0.74 mmol) and potassium carbonate (0.31 g, 2.22 mmol) to give the title compound as a white solid (0.12 g): MS (m/e): 441(M+1).

Provenance & Evidence