3-Aminophenylboronic acid → 3'-Amino-5-formyl-6-methoxy-biphenyl-3-sulfonamide

HRID 1454526Notes

Reaction equation

HRID 1454526 reaction equation
Br[C:2]1[CH:3]=[C:4]([S:12]([NH2:15])(=[O:14])=[O:13])[CH:5]=[C:6]([CH:10]=[O:11])[C:7]=1[O:8][CH3:9].[NH2:16][C:17]1[CH:18]=[C:19](B(O)O)[CH:20]=[CH:21][CH:22]=1>>[NH2:16][C:17]1[CH:22]=[C:21]([C:2]2[C:7]([O:8][CH3:9])=[C:6]([CH:10]=[O:11])[CH:5]=[C:4]([S:12]([NH2:15])(=[O:14])=[O:13])[CH:3]=2)[CH:20]=[CH:19][CH:18]=1

Participants

3

Reactant 2

HCID 922693-Aminophenylboronic acidHCID 866076983-Bromo-5-formyl-4-methoxy-benzenesulfonamide

Product 1

HCID 866077123'-Amino-5-formyl-6-methoxy-biphenyl-3-sulfonamide

Procedure

Proceeding as in Reference 19, but substituting 3-bromo-5-formyl-4-methoxy-benzenesulfonamide and 3-aminobenzene boronic acid, gave 3′-amino-5-formyl-6-methoxy-biphenyl-3-sulfonamide.

Sources & evidence

ORD record
ord-275032cff49a4b86afaa617ccad7f1f9
Source dataset
uspto-grants-2009_01
Patent number
US07479502B2

Reaction notes

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