1H-Pyrazole, 4-bromo-1-methyl- → HCID 66765337, compound

HRID 1466836Notes

Reaction equation

HRID 1466836 reaction equation
[CH2:1]([O:3][C:4](=[O:26])[CH2:5][C:6]1[CH:11]=[CH:10][C:9]([O:12][CH3:13])=[C:8]([S:14][C:15]2[C:23]3[C:18](=[CH:19][C:20]([Cl:24])=[CH:21][CH:22]=3)[NH:17][C:16]=2[CH3:25])[CH:7]=1)[CH3:2].Br[C:28]1[CH:29]=[N:30][N:31]([CH3:33])[CH:32]=1>>[CH2:1]([O:3][C:4](=[O:26])[CH2:5][C:6]1[CH:11]=[CH:10][C:9]([O:12][CH3:13])=[C:8]([S:14][C:15]2[C:23]3[C:18](=[CH:19][C:20]([Cl:24])=[CH:21][CH:22]=3)[N:17]([C:28]3[CH:29]=[N:30][N:31]([CH3:33])[CH:32]=3)[C:16]=2[CH3:25])[CH:7]=1)[CH3:2]

Participants

3

Reactant 2

HCID 1674331H-Pyrazole, 4-bromo-1-methyl-HCID 66765306HCID 66765306, compound

Product 1

HCID 66765337HCID 66765337, compound

Procedure

Prepared according to the procedure described in Example 42, Step 4, using the following starting materials: [3-(6-chloro-2-methyl-1H-indol-3-ylsulfanyl)-4-methoxy-phenyl]-acetic acid ethyl ester and 4-bromo-1-methylpyrazole.

Workup

  1. customPrepared

Sources & evidence

ORD record
ord-cb214c643c68415a8acdc404158cab48
Source dataset
uspto-grants-2015_04
Patent number
US09000025B2

Reaction notes

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