Trifluoroacetic acid → N-(4-(3-fluorophenyl)piperidin-3-yl)-3-(pyridin-4-yl)-1H-indazole-5-carboxamide

Participants

Reaction Steps

Trifluoroacetic acid (1 mL) was added to tert-butyl 4-(3-fluorophenyl)-3-(3-(pyridin-4-yl)-1-trityl-1H-indazole-5-carboxamido)piperidine-1-carboxylate (0.105 mmol). The reaction was stirred at room temperature for 30 minutes. Triethylsilane (1 drop) was added to the reaction and stirred for an additional 5 minutes. The reaction was concentrated in vacuo and purified using prep LC/MS.

Provenance & Evidence