Cyclopropylamine → HCID 63718779, compound

HRID 1467968Notes

Reaction equation

[NH:1]1[C:9]2[C:4](=[CH:5][C:6]([C:10]([OH:12])=O)=[CH:7][CH:8]=2)[CH:3]=[CH:2]1.[CH:13]1([NH2:16])[CH2:15][CH2:14]1>>[CH:13]1([NH:16][C:10]([C:6]2[CH:5]=[C:4]3[C:9](=[CH:8][CH:7]=2)[NH:1][CH:2]=[CH:3]3)=[O:12])[CH2:15][CH2:14]1

Participants

Reactant 2

HCID 69828Cyclopropylamine

HCID 742801H-Indole-5-Carboxylic Acid

Product 1

HCID 63718779HCID 63718779, compound

Procedure

The title compound was prepared by following the similar procedure as described in Intermediate-10, using 1H-indole-5-carboxylic acid and cyclopropanamine (0.34 g, 92%); MS: 201.1 (M+1).

Sources & evidence

ORD record: ord-3c80dd76af3f4bf2857ac13c81118b83
Source dataset: uspto-grants-2015_04
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US09000175B2

Reaction notes

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