5-Methoxyindole → HCID 67808965, compound

HRID 1468049Notes

Reaction equation

HRID 1468049 reaction equation
Cl[C:2]1[N:7]=[CH:6][C:5]([O:8][CH:9]2[CH2:14][CH2:13][N:12]([C:15]([O:17][C:18]([CH3:21])([CH3:20])[CH3:19])=[O:16])[CH2:11][CH2:10]2)=[CH:4][CH:3]=1.[CH3:22][O:23][C:24]1[CH:25]=[C:26]2[C:30](=[CH:31][CH:32]=1)[NH:29][CH:28]=[CH:27]2>>[C:18]([O:17][C:15]([N:12]1[CH2:13][CH2:14][CH:9]([O:8][C:5]2[CH:6]=[N:7][C:2]([N:29]3[C:30]4[C:26](=[CH:25][C:24]([O:23][CH3:22])=[CH:32][CH:31]=4)[CH:27]=[CH:28]3)=[CH:3][CH:4]=2)[CH2:10][CH2:11]1)=[O:16])([CH3:21])([CH3:20])[CH3:19]

Participants

3

Reactant 2

HCID 138725-MethoxyindoleHCID 86696180Tert-butyl 4-((6-chloropyridin-3-yl)oxy)piperidine-1-carboxylate

Product 1

HCID 67808965HCID 67808965, compound

Procedure

The title compound was prepared by following the similar procedure as described in Example-1 using tert-butyl 4-((6-chloropyridin-3-yl)oxy)piperidine-1-carboxylate (intermediate-06) and 5-methoxy-1H-indole (0.085 g, 20%).

Sources & evidence

ORD record
ord-6964fa2873c54d14bdc1b3ac5c280272
Source dataset
uspto-grants-2015_04
Patent number
US09000175B2

Reaction notes

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