2-Bromopyridine → HCID 68489605, compound

Participants

Reaction Conditions

Reaction Steps

Following the general procedure for the synthesis of 2-R-5-(heteroaryl-2-ylamino)phenol, 2-bromopyridine (0.6 mL, 6.33 mmol) and 5-amino-o-cresol (390 mg, 3.16 mmol) in 10% aqueous EtOH (10 mL) was heated at 90° C. for 18 h. The title compound was obtained after purification by flash chromatography on silica gel (hexane:EtOAc 6/4) in 43% yield (271 mg).

Provenance & Evidence