HRID1480278

反应详情

EQUATION

反应方程式

HRID 1480278 的结构方程式

PROCEDURE

实验过程

The title compound was synthesized in analogy to Example 112e, using 2-[[5-cyclopropyl-4-[(1S)-2,2,2-trifluoro-1-methyl-ethoxy]pyridine-2-carbonyl]amino]-3,3-dimethyl-butanoic acid (Example 199b) and 3,3-Difluoroazetidine hydrochloride (CAN 288315-03-7) as starting materials and isolated (35 mg, 58%); MS (ESI, m/z): 464.6 (M+H+).

WORKUP

后处理

  1. customisolated (35 mg, 58%)