HRID1480329

反应详情

EQUATION

反应方程式

HRID 1480329 的结构方程式

PROCEDURE

实验过程

The title compound was synthesized in analogy to Example 112e, using 5-(3,3-difluoroazetidin-1-yl)-4-(2,2,2-trifluoroethoxy)pyridine-2-carboxylic acid (example 223b) and 3-amino-3-cyclopropyl-butanamide (example 270c) as starting materials and isolated (70 mg, 63%) as a racemate; MS (ESI, m/z): 437.3 (M+H+).

WORKUP

后处理

  1. customisolated (70 mg, 63%) as a racemate