2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline → HCID 89996034, compound

HRID 1480848Notes

Reaction equation

HRID 1480848 reaction equation
[CH3:1][O:2][C:3]1[CH:9]=[C:8](B2OC(C)(C)C(C)(C)O2)[CH:7]=[CH:6][C:4]=1[NH2:5].Br[C:20]1[N:24]([CH2:25][CH2:26][O:27][CH3:28])[C:23]([CH3:29])=[N:22][CH:21]=1>>[CH3:1][O:2][C:3]1[CH:9]=[C:8]([C:20]2[N:24]([CH2:25][CH2:26][O:27][CH3:28])[C:23]([CH3:29])=[N:22][CH:21]=2)[CH:7]=[CH:6][C:4]=1[NH2:5]

Participants

3

Reactant 2

HCID 177502072-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)anilineHCID 89995732HCID 89995732, compound

Product 1

HCID 89996034HCID 89996034, compound

Procedure

The title compound was prepared according to the method described for Preparation 158 using 2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline and 5-bromo-1-(2-methoxyethyl)-2-methyl-1H-imidazole (Preparation 209).

Sources & evidence

ORD record
ord-888956f60351439eb0065b994e00182f
Source dataset
uspto-grants-2016_08
Patent number
US09409907B2

Reaction notes

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