1-Methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole → HCID 81288941, compound

HRID 1480852Notes

Reaction equation

HRID 1480852 reaction equation
Br[C:2]1[CH:8]=[CH:7][C:5]([NH2:6])=[C:4]([CH2:9][CH3:10])[CH:3]=1.[CH3:11][N:12]1[CH:16]=[C:15](B2OC(C)(C)C(C)(C)O2)[CH:14]=[N:13]1>>[CH2:9]([C:4]1[CH:3]=[C:2]([C:15]2[CH:14]=[N:13][N:12]([CH3:11])[CH:16]=2)[CH:8]=[CH:7][C:5]=1[NH2:6])[CH3:10]

Participants

3

Reactant 2

HCID 27739871-Methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazoleHCID 28012834-Bromo-2-ethylaniline

Product 1

HCID 81288941HCID 81288941, compound

Procedure

The title compound was prepared according to the method described for Preparation 98 using 4-bromo-2-ethylaniline and 1-methylpyrazole-4-boronic acid pinacol ester.

Sources & evidence

ORD record
ord-c158b8a2e9244cc28668de5e7f5ab285
Source dataset
uspto-grants-2016_08
Patent number
US09409907B2

Reaction notes

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