HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
3-Acetylphenylboronic acid → 1-(3-{2-[2-(4-Hydroxy-phenyl)-ethylamino]-pyrimidin-4-yl}-phenyl)-ethanone
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | 3-Acetylphenylboronic acid | HCID 2734310 | — |
| Edukt | 4-[2-(4-Chloro-pyrimidin-2-ylamino)-ethyl]-phenol | HCID 86603281 | — |
| Produkt | 1-(3-{2-[2-(4-Hydroxy-phenyl)-ethylamino]-pyrimidin-4-yl}-phenyl)-ethanone | HCID 67044689 | — |
Reaktionsschritte
Intermediate 61 was coupled with 3-acetyl phenylboronic acid following procedure A. LC-MS showed the product had the expected M+H+ of 334.
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US07732444B2 |
| Quelldatensatz | uspto-grants-2010_06 |
| ORD ID | ord-ed692131011341e3832ce46587a68031 |
| Quellennotiz | uspto-grants-2010_06 |