1-Methylindole → 1-Methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

HRID 1490476Notes

Reaction equation

HRID 1490476 reaction equation
Cn1ccc2ccccc21>CC1(C)OBOC1(C)C.[CH2-][Co+]12<-[N](=C(C)c3cccc(C(C)=[N]->1C1CCCCC1)[n]->23)C1CCCCC1>Cn1c(B2OC(C)(C)C(C)(C)O2)cc2ccccc21

Participants

4

Reactant 1

HCID 117811-Methylindole

Product 1

HCID 248855611-Methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indoleYield 59%

Reagents, catalysts & solvents 2

HCID 27347684,4,5,5-Tetramethyl[1,3,2]dioxaborolaneReagentHCID 178477760HCID 178477760, compoundCatalyst

Conditions

Temperature
80 °C

Sources & evidence

ORD record
ord-007e4516c96b4fe39eecc394269f1434
Source dataset
Borylation dataset from Roche

Reaction notes

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