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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1490573Generated: October 30, 2026

5-Methoxy-2-methylindole → 5-Methoxy-2-methyl-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

https://huagongshe.com/reaction/1490573

Reaction equation

Participants

RoleNameHCIDCharge
Reactant5-Methoxy-2-methylindoleHCID 70642—
Reagent4,4,5,5-Tetramethyl[1,3,2]dioxaborolaneHCID 2734768—
Reagent4,4'-Di-tert-butyl-2,2'-bipyridylHCID 4249187—
CatalystBis(1,5-cyclooctadiene)dimethoxydiiridiumHCID 76001521—
SolventHexaneHCID 8058—
Product5-Methoxy-2-methyl-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indoleHCID 2496059695%

Reaction Conditions

Temperature60 °C

Provenance & Evidence

DOI10.1021/ja0631652
Source datasetBorylation dataset from Roche
ORD IDord-eddc97ef822643a69559450057763888
Source noteBorylation dataset from Roche