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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1490580Generated: October 30, 2026

Ethyl 5-methoxyindole-2-carboxylate → Ethyl 5-methoxy-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-2-carboxylate

https://huagongshe.com/reaction/1490580

Reaction equation

Participants

RoleNameHCIDCharge
ReactantEthyl 5-methoxyindole-2-carboxylateHCID 20926—
Reagent4,4,5,5-Tetramethyl[1,3,2]dioxaborolaneHCID 2734768—
Reagent4,4'-Di-tert-butyl-2,2'-bipyridylHCID 4249187—
CatalystBis(1,5-cyclooctadiene)dimethoxydiiridiumHCID 76001521—
SolventHexaneHCID 8058—
ProductEthyl 5-methoxy-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-2-carboxylateHCID 2496059882%

Reaction Conditions

Temperature60 °C

Provenance & Evidence

DOI10.1021/ja0631652
Source datasetBorylation dataset from Roche
ORD IDord-acfe026613964bcfaefa7c284a88b1cd
Source noteBorylation dataset from Roche