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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1490581Generated: November 1, 2026

methyl 4-methoxy-1H-indole-2-carboxylate → Methyl 4-methoxy-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-2-carboxylate

https://huagongshe.com/reaction/1490581

Reaction equation

Participants

RoleNameHCIDCharge
Reactantmethyl 4-methoxy-1H-indole-2-carboxylateHCID 688172—
Reagent4,4,5,5-Tetramethyl[1,3,2]dioxaborolaneHCID 2734768—
Reagent4,4'-Di-tert-butyl-2,2'-bipyridylHCID 4249187—
CatalystBis(1,5-cyclooctadiene)dimethoxydiiridiumHCID 76001521—
SolventHexaneHCID 8058—
ProductMethyl 4-methoxy-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-2-carboxylateHCID 5343693479%

Reaction Conditions

Temperature60 °C

Provenance & Evidence

DOI10.1021/ja0631652
Source datasetBorylation dataset from Roche
ORD IDord-9fccf3a399154e63a7c61b5aee5146a1
Source noteBorylation dataset from Roche