HCID 89924094, compound → HCID 72948169, compound

HRID 1500901Notes

Reaction equation

HRID 1500901 reaction equation
[Cl:1][C:2]1[CH:20]=[CH:19][C:5]2[N:6]([C:11]3[CH:12]=[N:13][C:14]([O:17][CH3:18])=[CH:15][CH:16]=3)[C:7]([CH2:9]Cl)=[N:8][C:4]=2[CH:3]=1.[CH3:21][S:22]([C:25]1[C:33]2[C:28](=[CH:29][CH:30]=[CH:31][CH:32]=2)[NH:27][N:26]=1)(=[O:24])=[O:23]>>[Cl:1][C:2]1[CH:20]=[CH:19][C:5]2[N:6]([C:11]3[CH:12]=[N:13][C:14]([O:17][CH3:18])=[CH:15][CH:16]=3)[C:7]([CH2:9][N:27]3[C:28]4[C:33](=[CH:32][CH:31]=[CH:30][CH:29]=4)[C:25]([S:22]([CH3:21])(=[O:23])=[O:24])=[N:26]3)=[N:8][C:4]=2[CH:3]=1

Participants

3

Reactant 2

HCID 89924094HCID 89924094, compoundHCID 1785048563-methanesulfonyl-1H-indazole2×

Product 1

HCID 72948169HCID 72948169, compound

Procedure

The title compound was prepared in analogy to Example 3-1 by using 5-chloro-2-chloromethyl-1-(6-methoxy-pyridin-3-yl)-1H-benzoimidazole and 3-methanesulfonyl-1H-indazole instead of 5-chloro-2-chloromethyl-1-(4,4,4-tri fluoro-butyl)-1H-benzoimidazole and 3-methanesulfonyl-1H-indazole.

Sources & evidence

ORD record
ord-ab0b93c128be4a6e80ba2e0f94c38555
Source dataset
uspto-grants-2015_12
Patent number
US09206191B2

Reaction notes

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