HCID 22933768, compound → HCID 72948170, compound

HRID 1500902Notes

Reaction equation

HRID 1500902 reaction equation
[Cl:1][C:2]1[CH:19]=[CH:18][C:5]2[N:6]([C:11]3[CH:12]=[N:13][C:14]([Cl:17])=[CH:15][CH:16]=3)[C:7]([CH2:9]Cl)=[N:8][C:4]=2[CH:3]=1.CS(N1C2C(=CC=CC=2)C=N1)(=O)=O.[CH3:33][S:34]([C:37]1[C:45]2[C:40](=[CH:41][CH:42]=[CH:43][CH:44]=2)[NH:39][N:38]=1)(=[O:36])=[O:35]>>[Cl:1][C:2]1[CH:19]=[CH:18][C:5]2[N:6]([C:11]3[CH:12]=[N:13][C:14]([Cl:17])=[CH:15][CH:16]=3)[C:7]([CH2:9][N:39]3[C:40]4[C:45](=[CH:44][CH:43]=[CH:42][CH:41]=4)[C:37]([S:34]([CH3:33])(=[O:35])=[O:36])=[N:38]3)=[N:8][C:4]=2[CH:3]=1

Participants

4

Reactant 3

HCID 22933768HCID 22933768, compoundHCID 89924292HCID 89924292, compoundHCID 1785048563-methanesulfonyl-1H-indazole

Product 1

HCID 72948170HCID 72948170, compound

Procedure

The title compound was prepared in analogy to Example 3-1 by using 5-chloro-2-chloromethyl-1-(6-chloro-pyridin-3-yl)-1H-benzoimidazole and methanesulfonyl-1H-indazole instead of 5-chloro-2-chloromethyl-1-(4,4,4-trifluoro-butyl)-1H-benzoimidazole and 3-methanesulfonyl-1H-indazole.

Sources & evidence

ORD record
ord-106a178faca24d2a99dc91a1a0fe056d
Source dataset
uspto-grants-2015_12
Patent number
US09206191B2

Reaction notes

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