Cesium fluoride → HCID 11191016, compound

Participants

Reaction Steps

Using the procedure demonstrated in Example 9, react trifluoromethanesulfonic acid 6-methoxy-1-[4-(2-piperidin-1-yl-ethoxy)-phenoxy]-naphthalen-2-yl ester (800 mg, 1.52 mmol), 2,3-difluorobenzene boronic acid (720 mg, 4.57 mmol), cesium fluoride (2.1 g, 13.7 mmol), palladium(II)acetate (34 mg, 0.15 mmol) and tricyclohexylphosphine (64 mg, 0.23 mmol) to obtain 622 mg (84%) of the title compound: mass spectrum (ion spray) 490.4 (M+H).

Provenance & Evidence