反应详情

In analogy to the procedure described for the preparation of intermediate 1A, [6-chloro-3-methyl-5-(3-trifluoromethyl-phenyl)-pyridin-2-yl]-(4-pyrrolidin-1-yl-piperidin-1-yl)-methanone (example 3) was reacted with 5-(5,5-dimethyl-[1,3,2]dioxaborinan-2-yl)-1-methyl-1H-pyrazole to give the title compound as dark brown oil. MS: 498.2 (MH+).