HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-(3-{[(Benzyloxy)carbonyl]amino}oxetan-3-yl)acetic acid → 2-Oxo-2-[4-(pentafluoro-lambda6-sulfanyl)phenyl]ethyl (3-{[(benzyloxy)carbonyl]amino}oxetan-3-yl)acetate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-(3-{[(Benzyloxy)carbonyl]amino}oxetan-3-yl)acetic acid | HCID 89525437 | — |
| Reactant | 2-Bromo-1-[4-(pentafluoro-lambda6-sulfanyl)phenyl]ethanone | HCID 117601242 | — |
| Product | 2-Oxo-2-[4-(pentafluoro-lambda6-sulfanyl)phenyl]ethyl (3-{[(benzyloxy)carbonyl]amino}oxetan-3-yl)acetate | HCID 131733120 | — |
Reaction Steps
Prepared by Method E using (3-{[(benzyloxy)carbonyl]amino}oxetan-3-yl)acetic acid (Preparation 25, 0.647 g, 2.44 mmol) and 2-bromo-1-[4-(pentafluoro-λ6-sulfanyl)phenyl]-ethanone (Preparation 40, 0.793 g, 2.44 mmol) to afford the title compound.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09079878B2 |
| Source dataset | uspto-grants-2015_07 |
| ORD ID | ord-b96427a15bfc46db898487a9dcf54de2 |
| Source note | uspto-grants-2015_07 |