3-Chloro-6-iodopyridazine → HCID 86696138, compound

Participants

Reaction Steps

The title compound was prepared from (S)-6-(2-hydroxy-2-methylpropyl)-6-phenyl-3-{(S)-1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-ethyl}-1,3-oxazinan-2-one and 3-chloro-6-iodo-pyridazine following a procedure analogous to that described in Example 1. Yield: 62% of theory; LC (method 1): tR=1.88 min; Mass spectrum (ESI+): m/z=466/468 (Cl) [M+H]+.

Provenance & Evidence