3-Carboxyphenylboronic acid → HCID 66578424, compound

HRID 1528692Notes

Reaction equation

HRID 1528692 reaction equation
[CH2:1]([NH:8][C:9]([NH:11][C:12]1[C:13]([CH3:24])=[N:14][O:15][C:16]=1[C:17]1[CH:22]=[CH:21][C:20](Br)=[CH:19][CH:18]=1)=[O:10])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.[C:25]([C:28]1[CH:29]=[C:30](B(O)O)[CH:31]=[CH:32][CH:33]=1)([OH:27])=[O:26]>>[CH2:1]([NH:8][C:9](=[O:10])[NH:11][C:12]1[C:13]([CH3:24])=[N:14][O:15][C:16]=1[C:17]1[CH:22]=[CH:21][C:20]([C:32]2[CH:31]=[CH:30][CH:29]=[C:28]([C:25]([OH:27])=[O:26])[CH:33]=2)=[CH:19][CH:18]=1)[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 27339573-Carboxyphenylboronic acidHCID 66578576HCID 66578576, compound

Product 1

HCID 66578424HCID 66578424, compound

Procedure

Prepared according to the procedure described in Example 1, Step 7, using 1-benzyl-3-[5-(4-bromo-phenyl)-3-methyl-isoxazol-4-yl]-urea and 3-carboxyphenylboronic acid.

Workup

  1. customPrepared

Sources & evidence

ORD record
ord-948acdfcd1de4c23b9f2ed778ef62b91
Source dataset
uspto-grants-2015_07
Patent number
US09090573B2

Reaction notes

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