1267337-78-9 → HCID 66578650, compound

HRID 1529039Notes

Reaction equation

Br[C:2]1[CH:3]=[C:4]([CH:12]=[CH:13][CH:14]=1)[CH2:5][C:6]1([C:9]([OH:11])=[O:10])[CH2:8][CH2:7]1.[CH3:15][C:16]1[C:20]([CH:21]([OH:31])[CH2:22][CH2:23][CH2:24][C:25]2[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=2)=[C:19]([C:32]2[CH:37]=[CH:36][C:35](B3OC(C)(C)C(C)(C)O3)=[CH:34][CH:33]=2)[O:18][N:17]=1>>[OH:31][CH:21]([C:20]1[C:16]([CH3:15])=[N:17][O:18][C:19]=1[C:32]1[CH:33]=[CH:34][C:35]([C:2]2[CH:14]=[CH:13][CH:12]=[C:4]([CH2:5][C:6]3([C:9]([OH:11])=[O:10])[CH2:8][CH2:7]3)[CH:3]=2)=[CH:36][CH:37]=1)[CH2:22][CH2:23][CH2:24][C:25]1[CH:30]=[CH:29][CH:28]=[CH:27][CH:26]=1

Participants

Reactant 2

HCID 658153371267337-78-9

HCID 66578361HCID 66578361, compound

Product 1

HCID 66578650HCID 66578650, compound

Procedure

Prepared according to the procedure described in Example 1, Step 7, using 1-(3-bromo-benzyl)-cyclopropanecarboxylic acid and 1-{3-methyl-5-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]isoxazol-4-yl}-4-phenyl-butan-1-ol.

Workup

customPrepared

Sources & evidence

ORD record: ord-dbf07c55a5aa48d99db45779e8e3a9f3
Source dataset: uspto-grants-2015_07
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US09090573B2

Reaction notes

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