N-(tert-butoxycarbonyl)glycine → HCID 131726664, compound

Participants

Reaction Steps

(1S)-1-{5-[4-(4-diisopropylcarbamoyl-2-methoxy-phenoxy)-butoxy]-benzo[d]isoxazole-3-ylcarbamoyl}-2-phenyl-ethyl-ammonium methane sulfonic acid salt, the compound of EXAMPLE 3, was used as a starting material in place of {5-[4-(4-diisopropylcarbamoyl-2-methoxy-phenoxy)-butoxy]-benzo[d]isoxazole-3-ylcarbamoyl}-methyl-ammonium methane sulfonic acid used in the above EXAMPLE 6. According to the same method as in EXAMPLE 6, N-(t-butoxycarbonyl)glycine was used, the above title compound was obtained (yield: 80%).

Provenance & Evidence