Cyclopropylamine → 2-Cyclopropylamino-5-sulfamoylbenzoic acid

HRID 1608238Notes

Reaction equation

HRID 1608238 reaction equation
F[C:2]1[CH:10]=[CH:9][C:8]([S:11](=[O:14])(=[O:13])[NH2:12])=[CH:7][C:3]=1[C:4]([OH:6])=[O:5].[CH:15]1([NH2:18])[CH2:17][CH2:16]1>>[CH:15]1([NH:18][C:2]2[CH:10]=[CH:9][C:8]([S:11](=[O:14])(=[O:13])[NH2:12])=[CH:7][C:3]=2[C:4]([OH:6])=[O:5])[CH2:17][CH2:16]1

Participants

3

Reactant 2

HCID 69828CyclopropylamineHCID 24926842-Fluoro-5-sulfamoylbenzoic acid

Product 1

HCID 198486222-Cyclopropylamino-5-sulfamoylbenzoic acid

Procedure

The title compound is prepared from 2-fluoro-5-sulfamoylbenzoic acid and cyclopropylamine in substantially the same manner as in Reference Example 87.

Sources & evidence

ORD record
ord-69ac9c265e054a42a6ec193baf2627f7
Source dataset
uspto-grants-1989_09
Patent number
US04870074

Reaction notes

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