(Pyrimidin-5-yl)boronic acid → (NE)-N-[(3R)-3-(2-methylphenyl)-1-(2-methyl-4-pyridinyl)-3-(4-pyrimidin-5-ylphenyl)propylidene]hydroxylamine

Participants

Reaction Steps

In analogy to example 22, from (E,R)-3-(4-bromophenyl)-1-(2-methylpyridin-4-yl)-3-o-tolylpropan-1-one oxime (example 142, step 1) and pyrimidine-5-boronic acid was prepared the title compound as a white foam, MS (ESI+): m/z=409.3 ([M+H]+).

Provenance & Evidence