N-cyclopropyl-4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide → HCID 44250487, compound

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Obtained as a white solid (81%) as a single isomer (exact isomeric form not determined) from 6′-bromo-4-(2-morpholinoethoxy)spiro[cyclohexane-1,3′-indolin]-2′-one (preparation 27) and N-cyclopropyl-4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide (preparation 40) following the experimental procedure as described in preparation 38 followed by purification by flash chromatography (98:2 to 20:1 dichloromethane/methanol).

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