4-[5-(4-Methanesulfonylphenyl)-2,3-dihydrobenzofuran-2-yl]piperidine-1-carbonitrile → 4-[5-(4-Methanesulfonyl-phenyl)-2,3-dihydro-benzofuran-2-yl]-1-(3-propyl-[1,2,4]oxadiazol-5-yl)-piperidine

Participants

Reaction Steps

The title compound is prepared from 4-[5-(4-methanesulfonyl-phenyl)-2,3-dihydro-benzofuran-2-yl]-piperidine-1-carbonitrile and N-hydroxy-butyramidine following a procedure analogous to that described in Example 2. LC (method 2): tR=1.40 min; Mass spectrum (ESI+): m/z=468 [M+H]+.

Provenance & Evidence