HCID 70000726, compound → HCID 18678631, compound
Reaction equation
C(O[C:6](=O)[N:7]([C:9]1([S:15]([C:18]2[CH:23]=[CH:22][C:21]([C:24]3[N:28]=[C:27]([CH2:29][CH2:30][CH2:31][CH2:32][CH2:33][CH2:34][CH2:35][CH3:36])[O:26][N:25]=3)=[CH:20][CH:19]=2)(=[O:17])=[O:16])[CH2:14][CH2:13][NH:12][CH2:11][CH2:10]1)C)(C)(C)C>C(O)=O>[CH2:29]([C:27]1[O:26][N:25]=[C:24]([C:21]2[CH:22]=[CH:23][C:18]([S:15]([C:9]3([NH:7][CH3:6])[CH2:14][CH2:13][NH:12][CH2:11][CH2:10]3)(=[O:17])=[O:16])=[CH:19][CH:20]=2)[N:28]=1)[CH2:30][CH2:31][CH2:32][CH2:33][CH2:34][CH2:35][CH3:36]Participants
3
Reactant 1
Product 1
Reagents, catalysts & solvents 1
Procedure
A solution of (4-{[4-(5-octyl-1,2,4-oxadiazol-3-yl)phenyl]sulfonyl}-4-piperidinyl)-methylcarbamic acid t-butyl ester in formic acid was stirred at ambient temperature for 4 hours. Concentrated in vacuo to give 0.21 g of the product as a formate salt.
Workup
- concentrationConcentrated in vacuo
Sources & evidence
- ORD record
- ord-cc5dd177597c44338f3dbb83a7501f68
- Source dataset
- uspto-grants-2003_01
- Patent number
- US06506901B2
Reaction notes
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