Acetic Acid → HCID 59032966, compound

Participants

Reaction Steps

Prepared from N-[5-(2-amino-1-{R}-hydroxyethyl)-2-hydroxyphenyl]-methane-sulfonamide (0.136 g, 0.55 mmol), 3-[3-(4-{[4-formyl-1-piperidinyl]-sulfonyl}phenyl)-1,2,4-oxadiazol-5-yl]propanoic acid methyl ester (0.55 mmol), glacial acetic acid (0.040 g, 0.66 mmol) and sodium cyanoborohydride (0.0382 g, 0.061 mmol) according to the procedure used for example 67 (Step B) to give 0.180 g of the title compound as a white solid.

Provenance & Evidence