N-Hydroxyacetamidine → HCID 58002576, compound

Participants

Reaction Steps

100 mg (0.26 mmol) of the compound from Example 105A and 40 mg (0.534 mmol) of N′-hydroxyethanimidamide were reacted according to the General Method 2. Diastereomer separation of 62 mg of the cis/trans isomer mixture according to Method 12C gave 46 mg of the title compound and 5.7 mg of the trans isomer.

Provenance & Evidence