HCID 58989934, compound → HCID 58990026, compound

HRID 1663154Notes

Reaction equation

HRID 1663154 reaction equation
FC1C(O[C:9](=[O:24])[C:10]2[CH:15]=[CH:14][CH:13]=[CH:12][C:11]=2[NH:16][CH2:17][C:18]2[CH:23]=[CH:22][N:21]=[CH:20][CH:19]=2)=C(F)C(F)=C(F)C=1F.[CH2:29]([C:33]1[CH2:37][CH:36]([CH2:38][O:39][NH2:40])[O:35][N:34]=1)[CH2:30][CH2:31][CH3:32]>>[CH2:29]([C:33]1[CH2:37][CH:36]([CH2:38][O:39][NH:40][C:9](=[O:24])[C:10]2[CH:15]=[CH:14][CH:13]=[CH:12][C:11]=2[NH:16][CH2:17][C:18]2[CH:19]=[CH:20][N:21]=[CH:22][CH:23]=2)[O:35][N:34]=1)[CH2:30][CH2:31][CH3:32]

Participants

3

Reactant 2

HCID 58989934HCID 58989934, compoundHCID 58990003HCID 58990003, compound

Product 1

HCID 58990026HCID 58990026, compound

Procedure

Prepared by a similar method as described for example 415. Starting materials: 2-[(Pyridin-4-ylmethyl)-amino]-benzoic acid pentafluorophenyl ester (preparation 7C) and O-(3-butyl-4,5-dihydro-isoxazol-5-ylmethyl)-hydroxylamine (see preparation 91).

Workup

  1. customPrepared by a similar method

Sources & evidence

ORD record
ord-c07d240f44e84c55a57bd4e7a787d773
Source dataset
uspto-grants-2011_10
Patent number
US08034811B2

Reaction notes

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