Morpholine → HCID 58989842, compound

HRID 1663163Notes

Reaction equation

HRID 1663163 reaction equation
[CH:1]1([CH2:6][O:7][NH:8][C:9]([C:11]2[CH:16]=[CH:15][CH:14]=[CH:13][C:12]=2[NH:17][CH2:18][C:19]2[CH:20]=[CH:21][C:22]([F:28])=[C:23]([CH:27]=2)[C:24]([OH:26])=O)=[O:10])[CH2:5][CH2:4][CH2:3][CH2:2]1.[NH:29]1[CH2:34][CH2:33][O:32][CH2:31][CH2:30]1>>[CH:1]1([CH2:6][O:7][NH:8][C:9](=[O:10])[C:11]2[CH:16]=[CH:15][CH:14]=[CH:13][C:12]=2[NH:17][CH2:18][C:19]2[CH:20]=[CH:21][C:22]([F:28])=[C:23]([C:24]([N:29]3[CH2:34][CH2:33][O:32][CH2:31][CH2:30]3)=[O:26])[CH:27]=2)[CH2:5][CH2:4][CH2:3][CH2:2]1

Participants

3

Reactant 2

HCID 8083MorpholineHCID 58989765HCID 58989765, compound

Product 1

HCID 58989842HCID 58989842, compound

Procedure

Prepared by a similar procedure as described for the preparation of Example 499, starting from 5-[(2-cyclopentylmethoxycarbamoyl-phenylamino)methyl]-2-fluoro-benzoic acid (Example 496) and morpholine.

Workup

  1. customPrepared by a similar procedure
  2. customas described for the preparation of Example 499

Sources & evidence

ORD record
ord-18bebbc35a4f4704b67ab7b0c4218532
Source dataset
uspto-grants-2011_10
Patent number
US08034811B2

Reaction notes

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