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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1670022Generated: October 31, 2026

(2R)-N-methanesulfonyl-(4-chlorophenyl)alanine → 1-(1,1-Dimethylethyl) 1,2-aziridinedicarboxylate

https://huagongshe.com/reaction/1670022

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(2R)-N-methanesulfonyl-(4-chlorophenyl)alanineHCID 967528—
Reactant1-Tert-butyl 2-methyl aziridine-1,2-dicarboxylateHCID 11171653—
Product1-(1,1-Dimethylethyl) 1,2-aziridinedicarboxylateHCID 21025956—

Reaction Steps

The title compound was prepared following the procedure described in Step B of Intermediate 135 using methyl 1-BOC-2-aziridinecarboxylate prepared in Step B.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07989634B2
Source datasetuspto-grants-2011_08
ORD IDord-5fd1222b6cd146f39535fc8674f68235
Source noteuspto-grants-2011_08