1-(1,1-Dimethylethyl) 1,2-aziridinedicarboxylate → tert-Butyl 2-formylaziridine-1-carboxylate

HRID 1670023Notes

Reaction equation

HRID 1670023 reaction equation
CN1CCC[C@@H]1C=O.[C:9]([N:16]1[CH2:18][CH:17]1[C:19](O)=[O:20])([O:11][C:12]([CH3:15])([CH3:14])[CH3:13])=[O:10]>>[C:9]([N:16]1[CH2:18][CH:17]1[CH:19]=[O:20])([O:11][C:12]([CH3:15])([CH3:14])[CH3:13])=[O:10]

Participants

3

Reactant 2

HCID 210259561-(1,1-Dimethylethyl) 1,2-aziridinedicarboxylateHCID 53829762(2R)-1-methylpyrrolidine-2-carbaldehyde

Product 1

HCID 75068696tert-Butyl 2-formylaziridine-1-carboxylate

Procedure

The title compound was prepared following the procedure described in Intermediate 138 using 1-BOC-aziridine-2-carboxylic acid.

Sources & evidence

ORD record
ord-51d07f9af1094d059de5526dd2f87526
Source dataset
uspto-grants-2011_08
Patent number
US07989634B2

Reaction notes

Loading…