Benzenesulfonyl chloride → HCID 16125108, compound

HRID 1674699Notes

Reaction equation

HRID 1674699 reaction equation
[CH3:1][C:2]1([CH3:16])[C:6]([CH3:8])([CH3:7])[O:5][B:4]([C:9]2[CH:14]=[CH:13][C:12]([NH2:15])=[CH:11][CH:10]=2)[O:3]1.[C:17]1([S:23](Cl)(=[O:25])=[O:24])[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1>>[CH3:8][C:6]1([CH3:7])[C:2]([CH3:16])([CH3:1])[O:3][B:4]([C:9]2[CH:14]=[CH:13][C:12]([NH:15][S:23]([C:17]3[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=3)(=[O:25])=[O:24])=[CH:11][CH:10]=2)[O:5]1

Participants

3

Reactant 2

HCID 7369Benzenesulfonyl chlorideHCID 27346204-(Tetramethyl-1,3,2-dioxaborolan-2-yl)aniline

Product 1

HCID 16125108HCID 16125108, compound

Procedure

The following boronic acid pinacolate ester was prepared according to general procedure GP 4 from 4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenylamine and the appropriate phenyl sulfonyl chloride.

Sources & evidence

ORD record
ord-3c5eaff7d5f64a25a951065b77c83ee1
Source dataset
uspto-grants-2011_08
Patent number
US08003655B2

Reaction notes

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