1-Phenylcyclopropanecarboxylic acid → HCID 58696122, compound

HRID 1674701Notes

Reaction equation

HRID 1674701 reaction equation
[CH3:1][C:2]1([CH3:16])[C:6]([CH3:8])([CH3:7])[O:5][B:4]([C:9]2[CH:14]=[CH:13][C:12]([NH2:15])=[CH:11][CH:10]=2)[O:3]1.[C:17]1([C:23]2([C:26](O)=[O:27])[CH2:25][CH2:24]2)[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1>>[CH3:8][C:6]1([CH3:7])[C:2]([CH3:16])([CH3:1])[O:3][B:4]([C:9]2[CH:14]=[CH:13][C:12]([NH:15][C:26]([C:23]3([C:17]4[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=4)[CH2:25][CH2:24]3)=[O:27])=[CH:11][CH:10]=2)[O:5]1

Participants

3

Reactant 2

HCID 802061-Phenylcyclopropanecarboxylic acidHCID 27346204-(Tetramethyl-1,3,2-dioxaborolan-2-yl)aniline

Product 1

HCID 58696122HCID 58696122, compound

Procedure

Intermediate 26 was prepared in analogy to GP 5 by reaction of 4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenylamine with 1-phenyl-cyclopropanecarboxylic acid.

Sources & evidence

ORD record
ord-e71110328ddf4da6b77a4ed47ea2bdb0
Source dataset
uspto-grants-2011_08
Patent number
US08003655B2

Reaction notes

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