1H-Pyrazole-1-benzyl-4-boronic acid → HCID 67348260, compound

Participants

Reaction Steps

Prepared from 3-fluoro-4-(2-iodothieno[3,2-b]pyridin-7-yloxy)benzenamine (Example 6, Step A; 0.300 g, 0.777 mmol) and 4-((1H-pyrazol-1-yl)methyl)phenylboronic acid (0.196 g, 0.971 mmol) using the procedure described for Example 94, Step A, to provide the product (210 mg, 36%) as a brown solid. LRMS (esi+) m/e 417 (M+1) detected.

Provenance & Evidence