HRID1678412

反应详情

EQUATION

反应方程式

HRID 1678412 的结构方程式

CONDITIONS

反应条件

温度
80 °C

PROCEDURE

实验过程

Approximately half of the suspension prepared in step c was treated with (2R)-2-phenylpropylamine (1.16 mL, 8.14 mmol, 10.0 equiv). After heating to 80° C., the solvents were removed in vacuo, and the residue was purified by reverse-phase HPLC (Sunfire, 35-60% CH3CN/H2O, 0.1% TFA, 12 min) to afford 156 mg of the title compound. MS (ES+): m/e 528.1 [M+H]+.

WORKUP

后处理

  1. customthe solvents were removed in vacuo
  2. customthe residue was purified by reverse-phase HPLC (Sunfire, 35-60% CH3CN/H2O, 0.1% TFA, 12 min)