Benzyl Alcohol → HCID 178494001, compound

HRID 1679038Notes

Reaction equation

HRID 1679038 reaction equation
Cl[C:2]1[C:7]2[CH:8]=[N:9][C:10]3[NH:14][N:13]=[CH:12][C:11]=3[C:6]=2[N:5]2[N:15]=[CH:16][N:17]=[C:4]2[N:3]=1.ClC1C2C=NC3N(CC)N=CC=3C=2N2N=CN=C2N=1.C(O)[C:38]1[CH:43]=[CH:42][CH:41]=[CH:40][CH:39]=1.[CH2:45]([OH:47])C>>[C:38]1([C:2]2[C:7]3[CH:8]=[N:9][C:10]4[NH:14][N:13]=[CH:12][C:11]=4[C:6]=3[N:5]3[N:15]=[C:16]([O:47][CH3:45])[N:17]=[C:4]3[N:3]=2)[CH:43]=[CH:42][CH:41]=[CH:40][CH:39]=1

Participants

5

Reactant 4

HCID 244Benzyl AlcoholHCID 702EthanolHCID 227584865-Chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]-triazolo[1,5-a]pyrimidineHCID 178478325HCID 178478325, compound

Product 1

HCID 178494001HCID 178494001, compound

Procedure

By substituting the 5-chloro-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine of Example 15 for the 5-chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]Triazolo[1,5-a]pyrimidine and benzyl alcohol for the ethanol in the procedure of Example 4, 5-phenyl-methoxy-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine is obtained.

Sources & evidence

ORD record
ord-b22b6538f6dc4dc49327e3cb90f9e190
Source dataset
uspto-grants-1978_03
Patent number
US04078064

Reaction notes

Loading…