Ethynylpyridine → HCID 67263240, compound

Participants

Reaction Steps

3-((6-amino-5-bromopyridin-3-yl)methylamino)-N-cyclopropyl-4-fluorobenzamide (38 mg, 0.1 mmol) was reacted with 2-ethynylpyridine (0.1 mL) as described in procedure D of Example 5 to afford 3-((6-Amino-5-(2-(pyridin-2-yl)ethynyl)pyridin-3-yl)methylamino)-N-cyclopropyl-4-fluorobenzamide as a solid. It was used without further purification. LC/MS; (M+H)+=402.

Provenance & Evidence