Triethylamine → 4-{3-[2-(4-Chloro-phenyl)-2H-indazol-3-yl]-3-cyclohexyl-ureido}-3-methyl-benzoic acid methyl ester

Participants

Reaction Steps

In analogy to the procedure described in example 1.2, [2-(4-chloro-phenyl)-2H-indazol-3-yl]-cyclohexyl-amine (example 11.1) was reacted with 3-methyl-4-isocyanato-benzoic acid methyl ester (example 14.1) in 1,2-dichloroethane in the presence of Et3N (1.4 eq.) for 2 days under reflux conditions to give the title compound as brown solid. MS: m/e=517.1 [M+H+].

Provenance & Evidence