(2S)-2-[2-borono-4-(trifluoromethyl)phenoxy]-propanoic acid → HCID 11246757, compound

HRID 1694745Notes

Reaction equation

HRID 1694745 reaction equation
FC(F)(F)S(O[C:7]1[CH:12]=[CH:11][C:10]([S:13]([CH3:16])(=[O:15])=[O:14])=[CH:9][C:8]=1[F:17])(=O)=O.B([C:23]1[CH:34]=[C:33]([C:35]([F:38])([F:37])[F:36])[CH:32]=[CH:31][C:24]=1[O:25][C@@H:26]([CH3:30])[C:27]([OH:29])=[O:28])(O)O>>[F:17][C:8]1[CH:9]=[C:10]([S:13]([CH3:16])(=[O:14])=[O:15])[CH:11]=[CH:12][C:7]=1[C:31]1[CH:32]=[C:33]([C:35]([F:38])([F:37])[F:36])[CH:34]=[CH:23][C:24]=1[O:25][C@@H:26]([CH3:30])[C:27]([OH:29])=[O:28]

Participants

3

Reactant 2

HCID 67277101(2S)-2-[2-borono-4-(trifluoromethyl)phenoxy]-propanoic acidHCID 86006151HCID 86006151, compound

Product 1

HCID 11246757HCID 11246757, compound

Procedure

The title compound was prepared by the method of example 144 step (i) using the product from step (i) and the product from example 146 step (iv).

Sources & evidence

ORD record
ord-b5115e02e02f49cd80dd9f3c0c4aa9c4
Source dataset
uspto-grants-2012_04
Patent number
US08158820B2

Reaction notes

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