(2S)-2-(2-borono-4-chlorophenoxy)-propanoic acid → HCID 58333689, compound

HRID 1694752Notes

Reaction equation

HRID 1694752 reaction equation
B([C:4]1[CH:15]=[C:14]([Cl:16])[CH:13]=[CH:12][C:5]=1[O:6][C@@H:7]([CH3:11])[C:8]([OH:10])=[O:9])(O)O.FC(F)(F)S(O[C:23]1[CH:28]=[CH:27][C:26]([S:29]([CH3:32])(=[O:31])=[O:30])=[CH:25][C:24]=1[F:33])(=O)=O>>[Cl:16][C:14]1[CH:13]=[CH:12][C:5]([O:6][C@@H:7]([CH3:11])[C:8]([OH:10])=[O:9])=[C:4]([C:23]2[CH:28]=[CH:27][C:26]([S:29]([CH3:32])(=[O:31])=[O:30])=[CH:25][C:24]=2[F:33])[CH:15]=1

Participants

3

Reactant 2

HCID 67277298(2S)-2-(2-borono-4-chlorophenoxy)-propanoic acidHCID 86006151HCID 86006151, compound

Product 1

HCID 58333689HCID 58333689, compound

Procedure

The title compound was prepared by the method of example 155 using the product from example 151 step (iv) and the product from example 149 step (i).

Sources & evidence

ORD record
ord-9ccae3a7c2724d2bbd3e4447535f5a13
Source dataset
uspto-grants-2012_04
Patent number
US08158820B2

Reaction notes

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