N-Aminomorpholine → HCID 59568471, compound

Participants

Reaction Steps

As described for example 160c, 1-methyl-3-((5-methyl-3-(pyridin-2-yl)isoxazol-4-yl)methylamino)-1H-pyrazole-5-carboxylic acid (80 mg; 255 μmol) was converted, using 4-aminomorpholine instead of isopropylamine, to the title compound (101 mg, 71%) which was obtained as a white solid. MS: m/e=398.2 [M+H]+.

Provenance & Evidence